Tianeptine
Tianeptine是5-HT吸收选择性促进剂。
中文名：噻奈普汀
英文名：Tianeptine
CAS 号： 72797-41-2
分子式：C₂₁H₂₅ClN₂O₄S
分子量：436.95
纯度：>98.0%
| Description | Tianeptine is a selective facilitator of 5-HT uptake in vitro and in vivo. IC50 Value: N/A Target: 5-HT Receptor Tianeptine has no affinity for a wide range of receptors, including 5-HT and dopamine (IC50 > 10 μM) and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo. |
| Target | serotonin |
| References | [1]. Broqua P; Baudrie V; Chaouloff F Differential effects of the novel antidepressant tianeptine on L-5-hydroxytryptophan (5-HTP)-elicited corticosterone release and body weight loss. Eur Neuropsychopharmacol. 1992 Jun;2(2):115-20. |
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